编号:136472
CAS号:799841-81-9
三字母:H2N-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-CONH2
描 述:来源于 γ-2-MSH。γ-2-MSH 是一种 12 个氨基酸肽,为 POMC 的 N 末端片段,包含所有黑素皮质激素内源性激动剂配体共有的 His-Phe-Arg-Trp 构像。
编号:200256
CAS号:72629-65-3
三字母:H2N-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-CONH2
描 述:一种来源于ACTH 1-13的激素,是一种内源性黑素皮质素MC3受体激动剂(pKi=7.46),其选择性是MC4的约40倍。它刺激黑色素生成,促进学习和记忆,并可影响炎症和免疫反应以及外周神经再生。
编号:166784
CAS号:162558-08-9
三字母:H2N-Lys-Thr-Trp-Gly-Gln-Tyr-Trp-Gln-Val-OH
描 述:PMEL 17可能是一种黑色素生成酶。 该序列已被鉴定为gp100表位,该表位在体内HLA-A2中可被肿瘤浸润淋巴细胞(TIL)识别。
编号:143583
CAS号:181477-43-0
三字母:H2N-Ile-Met-Asp-Gln-Val-Pro-Phe-Ser-Val-OH
描 述:Modified sequence of the gp100 epitope gp(209-217) ITDQVPFSV, in which a methionine replaced the natural threonine at position 2, bound to the HLA-A2 molecule with greater affinity than the unmodified peptide and was shown to have an increased ability to
编号:189964
CAS号:121062-08-6
三字母:Ac-Nle-cyclo(Asp-His-DPhe-Arg-Trp-Lys-NH2)
描 述:Melanotan (MT)-II是一种合成的黑皮质素 (melanocortin) 受体激动剂。它是可注射用的多肽荷尔蒙,可促进晒黑。
编号:206329
CAS号:128315-56-0
三字母:H2N-Asp-Phe-Asp-Met-Leu-Arg-Cys-Met-Leu-Gly-Arg-Val-Tyr-Arg-Pro-Cys-Trp-Gln-Val-OH(Disulfide Bridge:Cys7-Cys16)
描 述:MCH是内源性黑色素浓度激素受体激动剂,在MCH1和MCH2受体处的IC50值分别为0.3和1.5nM。它可以增加体内的食物摄入量。
编号:143927
CAS号:162558-10-3
三字母:H2N-Ile-Thr-Asp-Gln-Val-Pro-Phe-Ser-Val-OH
描 述:As KTWGQYWQV, ITDQVPFSV is a gp100 epitope that is recognized in the context of HLA-A2 by tumor-infiltrating lymphocytes (TIL) in vivo. PMEL 17 could be a melanogenic enzyme.
编号:146674
CAS号:255710-51-1
三字母:H2N-Ile-Met-Gln-Val-Pro-Phe-Ser-Val-OH
描 述:
编号:180556
CAS号:319927-23-6
三字母:H2N-Ile-Thr-Gln-Val-Pro-Phe-Ser-Val-OH
描 述: