一种特定的caspase-3抑制剂。
编号：196099
CAS号：210344-95-9
单字母：Z-D(OMe)-E(OMe)-V-D(OMe)-FMK
| 编号: | 196099 |
| 中文名称: | 半胱氨酸蛋白酶Caspase-3 Inhibitor |
| CAS号: | 210344-95-9 |
| 单字母: | Z-D(OMe)-E(OMe)-V-D(OMe)-FMK |
| 三字母: | Cbz N端Cbz保护 -Asp(OMe)暂无说明 -Glu(OMe)暂无说明 -Val缬氨酸 -Asp(OMe)暂无说明 -FMKC端氟甲基酮修饰 |
| 氨基酸个数: | 4 |
| 分子式: | C30H41O12N4F1 |
| 平均分子量: | 668.66 |
| 精确分子量: | 668.27 |
| 等电点(PI): | - |
| pH=7.0时的净电荷数: | - |
| 平均亲水性: | -1.5 |
| 疏水性值: | 4.2 |
| 消光系数: | - |
| 来源: | 人工化学合成，仅限科学研究使用，不得用于人体。 |
| 盐体系: | 可选TFA、HAc、HCl或其它 |
| 储存条件: | 负80℃至负20℃ |
| 标签: | CBZ修饰肽 侧链保护基肽 FMK修饰肽 |
Methyl ester of Z-DEVD-FMK, a specific caspase-3 inhibitor. Z-D(OMe)E(OMe)VD(OMe)-FMK reduces vulnerability to the neuronal death that occurs in the aftermath of kainic acid-evoked status epilepticus (SE).
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